Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50002844
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463643BDBM50463643(CHEMBL4242974)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463649BDBM50463649(GSK-1292263A | GSK-263A | Gsk 1292263 | Gsk-129226...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463652BDBM50463652(CHEMBL4248331)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463637BDBM50463637(CHEMBL4240810)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463647BDBM50463647(CHEMBL4242383)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463641BDBM50463641(CHEMBL4239711)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463648BDBM50463648(CHEMBL4243608)
Affinity DataEC50:  147nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463651BDBM50463651(CHEMBL4243251)
Affinity DataEC50:  179nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463636BDBM50463636(CHEMBL4249284)
Affinity DataEC50:  345nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463638BDBM50463638(CHEMBL4248698)
Affinity DataEC50:  452nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463644BDBM50463644(CHEMBL4248913)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463650BDBM50463650(CHEMBL4239203)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463646BDBM50463646(CHEMBL4244903)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463639BDBM50463639(CHEMBL4244655)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29080BDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at GPR119 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463642BDBM50463642(CHEMBL4239244)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at GPR119 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463640BDBM50463640(CHEMBL4238669)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463645BDBM50463645(CHEMBL4249171)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells assessed as cAMP accumulation after 1 hr by ultra LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed