Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50003333
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31539BDBM31539(pyrazolo[4,3-h]quinazoline-3-carboxamide, 22)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31532BDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31539BDBM31539(pyrazolo[4,3-h]quinazoline-3-carboxamide, 22)
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31543BDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470534BDBM50470534(CHEMBL4288758)
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470534BDBM50470534(CHEMBL4288758)
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110183BDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31539BDBM31539(pyrazolo[4,3-h]quinazoline-3-carboxamide, 22)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31532BDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31543BDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470523BDBM50470523(CHEMBL4286430)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110183BDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470534BDBM50470534(CHEMBL4288758)
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470523BDBM50470523(CHEMBL4286430)
Affinity DataIC50: 26nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470535BDBM50470535(CHEMBL4289852)
Affinity DataIC50: 29nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470533BDBM50470533(CHEMBL4278514)
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470525BDBM50470525(CHEMBL4281557)
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470525BDBM50470525(CHEMBL4281557)
Affinity DataIC50: 34nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470535BDBM50470535(CHEMBL4289852)
Affinity DataIC50: 36nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31533BDBM31533(pyrazolo[4,3-h]quinazoline-3-carboxamide, 16)
Affinity DataIC50: 37nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470533BDBM50470533(CHEMBL4278514)
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470524BDBM50470524(CHEMBL4287981)
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470525BDBM50470525(CHEMBL4281557)
Affinity DataIC50: 45nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31532BDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)
Affinity DataIC50: 58nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470524BDBM50470524(CHEMBL4287981)
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470531BDBM50470531(CHEMBL4294798)
Affinity DataIC50: 120nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470519BDBM50470519(CHEMBL4292180)
Affinity DataIC50: 120nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31533BDBM31533(pyrazolo[4,3-h]quinazoline-3-carboxamide, 16)
Affinity DataIC50: 160nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470519BDBM50470519(CHEMBL4292180)
Affinity DataIC50: 250nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470520BDBM50470520(CHEMBL4283123)
Affinity DataIC50: 250nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31542BDBM31542(pyrazolo[4,3-h]quinazoline-3-carboxamide, 25)
Affinity DataIC50: 280nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470524BDBM50470524(CHEMBL4287981)
Affinity DataIC50: 320nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31542BDBM31542(pyrazolo[4,3-h]quinazoline-3-carboxamide, 25)
Affinity DataIC50: 330nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31542BDBM31542(pyrazolo[4,3-h]quinazoline-3-carboxamide, 25)
Affinity DataIC50: 350nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470520BDBM50470520(CHEMBL4283123)
Affinity DataIC50: 450nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470531BDBM50470531(CHEMBL4294798)
Affinity DataIC50: 450nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470519BDBM50470519(CHEMBL4292180)
Affinity DataIC50: 470nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110183BDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataIC50: 500nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470521BDBM50470521(CHEMBL4281978)
Affinity DataIC50: 550nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470527BDBM50470527(CHEMBL4293299)
Affinity DataIC50: 620nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470530BDBM50470530(CHEMBL4294376)
Affinity DataIC50: 650nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470521BDBM50470521(CHEMBL4281978)
Affinity DataIC50: 680nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470523BDBM50470523(CHEMBL4286430)
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470522BDBM50470522(CHEMBL4286071)
Affinity DataIC50: 830nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470535BDBM50470535(CHEMBL4289852)
Affinity DataIC50: 850nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470527BDBM50470527(CHEMBL4293299)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470533BDBM50470533(CHEMBL4278514)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31533BDBM31533(pyrazolo[4,3-h]quinazoline-3-carboxamide, 16)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470532BDBM50470532(CHEMBL4287560)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Jiangnan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470521BDBM50470521(CHEMBL4281978)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
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