Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50003296
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469157BDBM50469157(CHEMBL4284736)
Affinity DataIC50: 6nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469159BDBM50469159(CHEMBL4283840)
Affinity DataIC50: 17nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469154BDBM50469154(CHEMBL4283678)
Affinity DataIC50: 29nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469165BDBM50469165(CHEMBL4291540)
Affinity DataIC50: 41nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469162BDBM50469162(CHEMBL4282733)
Affinity DataIC50: 41nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469170BDBM50469170(CHEMBL4291025)
Affinity DataIC50: 42nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469166BDBM50469166(CHEMBL4294422)
Affinity DataIC50: 52nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469169BDBM50469169(CHEMBL4292925)
Affinity DataIC50: 72nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469164BDBM50469164(CHEMBL4287199)
Affinity DataIC50: 98nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469160BDBM50469160(CHEMBL4280386)
Affinity DataIC50: 104nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469167BDBM50469167(CHEMBL4279276)
Affinity DataIC50: 105nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469161BDBM50469161(CHEMBL4290610)
Affinity DataIC50: 107nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469163BDBM50469163(CHEMBL4282334)
Affinity DataIC50: 175nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469168BDBM50469168(CHEMBL4281328)
Affinity DataIC50: 225nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469156BDBM50469156(CHEMBL4291944)
Affinity DataIC50: 227nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469158BDBM50469158(CHEMBL4280228)
Affinity DataIC50: 495nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469155BDBM50469155(CHEMBL4288133)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed