Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50003120
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50467198(CHEMBL4287064)
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50467201(CHEMBL1470309)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50000541(Leutrol | CHEMBL93 | N-(1-Benzo(b)thien-2-ylethyl)...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50467199(CHEMBL1495111)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50467200(CHEMBL4286661)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM56424(4-methoxy-N-(1-piperidinylcarbonothioyl)benzamide ...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Vellore Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50467202(CHEMBL4284279)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human 5-LOX expressed in Escherichia coli BL21 using arachidonic acid as substrate by UV-vis spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed