Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50002334
TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021498(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021500(1N-[4-cyclopropylmethyl-10,17-dihydroxy-(13R,14R,1...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021495(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021493(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021498(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021499(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021499(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021495(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021493(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021495(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021493(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021499(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021490(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021498(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021502(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021500(1N-[4-cyclopropylmethyl-10,17-dihydroxy-(13R,14R,1...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021492(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021497(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021501(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021496(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021490(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  27nMAssay Description:Compound was tested for binding affinity against delta opioid receptor in guinea pig brain membrane using [3H]-EK as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021496(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021500(1N-[4-cyclopropylmethyl-10,17-dihydroxy-(13R,14R,1...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021497(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021491(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021502(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021504(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021494(1N-[10,17-dihydroxy-4-methyl-(13R,14R,17S)-12-oxa-...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021492(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021490(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021504(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021491(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021503(1N-[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12-oxa-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021501(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021492(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021501(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021497(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021502(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021503(1N-[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12-oxa-...)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021504(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021491(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50021494(1N-[10,17-dihydroxy-4-methyl-(13R,14R,17S)-12-oxa-...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021496(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021494(1N-[10,17-dihydroxy-4-methyl-(13R,14R,17S)-12-oxa-...)
Affinity DataKi:  4.40E+3nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50021503(1N-[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12-oxa-...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed