Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50002518
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459632(CHEMBL4204645)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459647(CHEMBL4205102)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459633(CHEMBL4205134)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459645(CHEMBL4213030)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459648(CHEMBL4210423)
Affinity DataIC50: 5nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459636(CHEMBL4205550)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459646(CHEMBL4211832)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459650(CHEMBL4217781)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459634(CHEMBL4216838)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459631(CHEMBL4212945)
Affinity DataIC50: 11nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459635(CHEMBL4207794)
Affinity DataIC50: 13nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50432829(CHEMBL2171700)
Affinity DataIC50: 31nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459643(CHEMBL4205210)
Affinity DataIC50: 38nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459644(CHEMBL4208034)
Affinity DataIC50: 44nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459638(CHEMBL4216917)
Affinity DataIC50: 47nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459641(CHEMBL4211452)
Affinity DataIC50: 53nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459637(CHEMBL4210880)
Affinity DataIC50: 140nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459649(CHEMBL4203751)
Affinity DataIC50: 380nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50432829(CHEMBL2171700)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459642(CHEMBL4217446)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459639(CHEMBL4208632)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459640(CHEMBL4211528)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMonoglyceride lipase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459640(CHEMBL4211528)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of His-tagged human MAGL expressed in Escherichia coli BL21(DE3) assessed as reduction in arachidonic acid production from 2-arachidonoylg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50459645(CHEMBL4213030)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human FAAH expressed in CHOK1 cells using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed