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Found 4 Enz. Inhib. hit(s) with all data for entry = 50002529
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50303803(1-((3aS,4R,9bR)-4-(6-bromobenzo[d][1,3]dioxol-5-yl...)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50459751(CHEMBL4212956)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50459750(CHEMBL4204670)
Affinity DataEC50:  480nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50459749(CHEMBL4204236)
Affinity DataEC50:  20nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed