TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University
Curated by ChEMBL
Saint Louis University
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University
Curated by ChEMBL
Saint Louis University
Curated by ChEMBL
Affinity DataEC50: 1.62E+3nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University
Curated by ChEMBL
Saint Louis University
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
Saint Louis University
Curated by ChEMBL
Saint Louis University
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair