Compile Data Set for Download or QSAR
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Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50002532
TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459795(CHEMBL4210443)
Affinity DataIC50:  15nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459793(CHEMBL4205572)
Affinity DataIC50:  19nMAssay Description:Displacement of biotinylated acetylated peptide from poly His-tagged CBP bromodomain (unknown origin) expressed in Escherichia coli BL21(DE3) by Alph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459791(CHEMBL4207490)
Affinity DataIC50:  40nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459792(CHEMBL4206032)
Affinity DataIC50:  59nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459798(CHEMBL4203144)
Affinity DataIC50:  140nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459790(CHEMBL4202606)
Affinity DataIC50:  146nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459797(CHEMBL4214796)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459789(CHEMBL4206088)
Affinity DataIC50:  7.70E+3nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459793(CHEMBL4205572)
Affinity DataKd:  35nMAssay Description:Displacement of biotinylated acetylated peptide from poly His-tagged CBP bromodomain (unknown origin) expressed in Escherichia coli BL21(DE3) measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459796(CHEMBL4210917)
Affinity DataKd:  2.00E+4nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459795(CHEMBL4210443)
Affinity DataKd:  3nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459799(CHEMBL4217805)
Affinity DataKd:  1.40E+3nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459792(CHEMBL4206032)
Affinity DataKd:  85nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459789(CHEMBL4206088)
Affinity DataKd:  970nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459788(CHEMBL4213403)
Affinity DataKd:  1.40E+3nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459794(CHEMBL4218324)
Affinity DataKd:  4.00E+3nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)