Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50003307 Sort by
TargetProstaglandin G/H synthase 1(Sheep)
Universidade Federal De Pernambuco (Ufpe)

Curated by ChEMBL
LigandPNGBDBM50469275(CHEMBL4290673)
Affinity DataIC50: 180nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Universidade Federal De Pernambuco (Ufpe)

Curated by ChEMBL
LigandPNGBDBM50469275(CHEMBL4290673)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human COX-2 expressed in Baculovirus infected Sf21 cells using arachidonic acid as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Universidade Federal De Pernambuco (Ufpe)

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human COX-2 expressed in Baculovirus infected Sf21 cells using arachidonic acid as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Universidade Federal De Pernambuco (Ufpe)

Curated by ChEMBL
LigandPNGBDBM50469276(CHEMBL4282782)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human COX-2 expressed in Baculovirus infected Sf21 cells using arachidonic acid as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Universidade Federal De Pernambuco (Ufpe)

Curated by ChEMBL
LigandPNGBDBM50469276(CHEMBL4282782)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Universidade Federal De Pernambuco (Ufpe)

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed