Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50003308
TargetFibroblast growth factor receptor 1(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322535BDBM50322535(3-[2-(Imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-meth...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322535BDBM50322535(3-[2-(Imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-meth...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469285BDBM50469285(CHEMBL4279567)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469288BDBM50469288(CHEMBL4290418)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469283BDBM50469283(CHEMBL4284111)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469279BDBM50469279(CHEMBL4283032)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469289BDBM50469289(CHEMBL4293500)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469281BDBM50469281(CHEMBL4287006)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469306BDBM50469306(CHEMBL4278749)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469290BDBM50469290(CHEMBL4287420)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469295BDBM50469295(CHEMBL4282621)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469287BDBM50469287(CHEMBL4294290)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469299BDBM50469299(CHEMBL4277682)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469300BDBM50469300(CHEMBL4287484)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469286BDBM50469286(CHEMBL4290903)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469277BDBM50469277(CHEMBL4281295)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469304BDBM50469304(CHEMBL4294291)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469301BDBM50469301(CHEMBL4286404)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469302BDBM50469302(CHEMBL4279766)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469280BDBM50469280(CHEMBL4289675)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469297BDBM50469297(CHEMBL4293899)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469278BDBM50469278(CHEMBL4289419)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469282BDBM50469282(CHEMBL4287074)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469292BDBM50469292(CHEMBL4277428)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469298BDBM50469298(CHEMBL4277269)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469296BDBM50469296(CHEMBL4285999)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428461BDBM50428461(CHEMBL2334797)
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469303BDBM50469303(CHEMBL4280203)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469305BDBM50469305(CHEMBL4290490)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428462BDBM50428462(CHEMBL2334796)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469294BDBM50469294(CHEMBL4279152)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469284BDBM50469284(CHEMBL4294709)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469291BDBM50469291(CHEMBL4284711)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469293BDBM50469293(CHEMBL4283719)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged human GSK-3beta expressed in Baculovirus infected SF9 cells using prephosphorylated-GS2 polype...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed