Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50008605
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520752BDBM50520752(CHEMBL4474261)
Affinity DataKi:  0.00800nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520751BDBM50520751(CHEMBL4473891)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520749BDBM50520749(CHEMBL4459250)
Affinity DataKi:  0.100nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520742BDBM50520742(CHEMBL4526105)
Affinity DataKi:  0.140nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520745BDBM50520745(CHEMBL4444395)
Affinity DataKi:  0.300nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520747BDBM50520747(CHEMBL4532723)
Affinity DataKi:  0.380nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520750BDBM50520750(CHEMBL4452621)
Affinity DataKi:  1.10nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520743BDBM50520743(CHEMBL4444545)
Affinity DataKi:  1.60nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520746BDBM50520746(CHEMBL4569180)
Affinity DataKi:  16nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520744BDBM50520744(CHEMBL4444772)
Affinity DataKi:  17nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520748BDBM50520748(CHEMBL4588251)
Affinity DataKi:  18nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520741BDBM50520741(CHEMBL4561948)
Affinity DataKi:  27nMAssay Description:Inhibition of HIV1 protease using fluorogenic substrate by continuous fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed