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Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50003315
TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469391(CHEMBL4288463)
Affinity DataEC50:  197nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50450236(Efatutazone)
Affinity DataEC50:  1nMAssay Description:Transactivation of PPARgamma (unknown origin) transfected in human DRO cells after 24 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469392(CHEMBL4289861)
Affinity DataEC50:  177nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469393(CHEMBL4281564)
Affinity DataEC50:  17nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469394(CHEMBL4286027)
Affinity DataEC50:  2.70nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469395(CHEMBL4277723)
Affinity DataEC50:  33nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469396(CHEMBL4282451)
Affinity DataEC50:  166nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469397(CHEMBL4277928)
Affinity DataEC50:  151nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50103521(Actos | CHEBI:8228 | Duetact | Pioglitazone | US10...)
Affinity DataEC50:  2.05E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50093473(Arhalofenate | CB-102 | JNJ-39659100 | M-102 | MBX...)
Affinity DataEC50:  7.37E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469398(ATx08-001 | FK-614)
Affinity DataEC50: >500nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as cell differentiation after 5 days by Hoechst 33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469399(CHEMBL4293061)
Affinity DataEC50:  57nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469398(ATx08-001 | FK-614)
Affinity DataEC50:  163nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469400(CHEMBL4278109)
Affinity DataEC50:  2.40nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50093473(Arhalofenate | CB-102 | JNJ-39659100 | M-102 | MBX...)
Affinity DataEC50: >500nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as cell differentiation after 5 days by Hoechst 33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469401(CHEMBL4289449)
Affinity DataEC50:  84nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469402(CHEMBL4288363)
Affinity DataEC50:  13nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469403(CHEMBL4285849)
Affinity DataEC50:  593nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50428854(CHEMBL1236924)
Affinity DataEC50: >500nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as cell differentiation after 5 days by Hoechst 33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469404(CHEMBL4279177)
Affinity DataEC50:  251nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50428854(CHEMBL1236924)
Affinity DataEC50:  59nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)