Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50003021
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465892BDBM50465892(CHEMBL3742031)
Affinity DataKi:  4nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465887BDBM50465887(CHEMBL4279554)
Affinity DataKi:  33nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465881BDBM50465881(CHEMBL4292785)
Affinity DataKi:  36nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465878BDBM50465878(CHEMBL4279370)
Affinity DataKi:  46nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465889BDBM50465889(CHEMBL4283935)
Affinity DataKi:  51nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465896BDBM50465896(CHEMBL4283888)
Affinity DataKi:  61nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465898BDBM50465898(CHEMBL4286216)
Affinity DataKi:  64nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465890BDBM50465890(CHEMBL4287299)
Affinity DataKi:  71nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465893BDBM50465893(CHEMBL4284942)
Affinity DataKi:  83nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465873BDBM50465873(CHEMBL4285967)
Affinity DataKi:  85nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465882BDBM50465882(CHEMBL4282181)
Affinity DataKi:  93nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465895BDBM50465895(CHEMBL4287182)
Affinity DataKi:  183nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465897BDBM50465897(CHEMBL4291161)
Affinity DataKi:  190nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465876BDBM50465876(CHEMBL4288719)
Affinity DataKi:  210nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465885BDBM50465885(CHEMBL4281515)
Affinity DataKi:  220nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465879BDBM50465879(CHEMBL4290711)
Affinity DataKi:  240nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465884BDBM50465884(CHEMBL4278060)
Affinity DataKi:  280nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465874BDBM50465874(CHEMBL4282584)
Affinity DataKi:  450nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465891BDBM50465891(CHEMBL4282823)
Affinity DataKi:  560nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465875BDBM50465875(CHEMBL4289377)
Affinity DataKi:  1.28E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465877BDBM50465877(CHEMBL4282120)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465888BDBM50465888(CHEMBL4290000)
Affinity DataKi:  2.54E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465886BDBM50465886(CHEMBL4276994)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465894BDBM50465894(CHEMBL4292140)
Affinity DataKi:  3.53E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465880BDBM50465880(CHEMBL4290457)
Affinity DataKi:  4.78E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGenome polyprotein(EV71)
Nankai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50465883BDBM50465883(CHEMBL4278711)
Affinity DataKi:  6.21E+3nMAssay Description:Inhibition of EV71 3C protease expressed in Escherichia coli BL21(DE3) using NMA-IEALFQGPPK(DNP)FR as substrate preincubated for 0.5 hrs followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed