Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50006834
TargetAndrogen receptor(Rat)
Southern Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503736BDBM50503736(CHEMBL4475784)
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Southern Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50425732BDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 1.32E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Southern Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503733BDBM50503733(CHEMBL4455261)
Affinity DataIC50: 3.66E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Southern Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503734BDBM50503734(CHEMBL4466881)
Affinity DataIC50: 3.82E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Southern Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503732BDBM50503732(CHEMBL4553704)
Affinity DataIC50: 4.03E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Southern Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50503735BDBM50503735(CHEMBL4476484)
Affinity DataIC50: 4.22E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed