Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50008344
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518343BDBM50518343(CHEMBL4519813)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50357312BDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518348BDBM50518348(CHEMBL4582434)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50460964BDBM50460964(CHEMBL4226237)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518344BDBM50518344(CHEMBL4444564)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518345BDBM50518345(CHEMBL4439998)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518342BDBM50518342(CHEMBL4541798)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518346BDBM50518346(CHEMBL4446870)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518347BDBM50518347(CHEMBL4514143)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518340BDBM50518340(CHEMBL4545868)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50518341BDBM50518341(CHEMBL4531607)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant full-length human N-terminal GST-fused BTK (2 to 659 residues) expressed in baculovirus expression system using biotin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed