Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50008364
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50161646((R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DOI from recombinant human 5HT2C receptor expressed in HEK293T cell membranes after 1 hr by beta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518473(CHEMBL4580763)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518478(CHEMBL4569512)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518478(CHEMBL4569512)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518473(CHEMBL4580763)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50161646((R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]DOI from recombinant human 5HT2A receptor expressed in HEK293T cell membranes after 1 hr by beta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50161646((R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]DOI from recombinant human 5HT2B receptor expressed in HEK293T cell membranes after 1 hr by beta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518479(CHEMBL4465663)
Affinity DataKi:  338nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518477(CHEMBL4482880)
Affinity DataKi:  343nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518473(CHEMBL4580763)
Affinity DataKi:  414nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518479(CHEMBL4465663)
Affinity DataKi:  422nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518479(CHEMBL4465663)
Affinity DataKi:  434nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518478(CHEMBL4569512)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518477(CHEMBL4482880)
Affinity DataKi:  552nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518477(CHEMBL4482880)
Affinity DataKi:  1.14E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518476(CHEMBL4436605)
Affinity DataKi:  2.31E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518476(CHEMBL4436605)
Affinity DataKi:  2.68E+3nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518475(CHEMBL4565350)
Affinity DataKi:  3.04E+3nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518475(CHEMBL4565350)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518476(CHEMBL4436605)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518474(CHEMBL4550346)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518474(CHEMBL4550346)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518472(CHEMBL4457398)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518472(CHEMBL4457398)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from 5HT2B receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518472(CHEMBL4457398)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518474(CHEMBL4550346)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50518475(CHEMBL4565350)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor (unknown origin) expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed