Compile Data Set for Download or QSAR
Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 50009708
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086170BDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataKi:  2nMAssay Description:Inhibition of human A2B adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531447BDBM50531447(CHEMBL4569909)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531478BDBM50531478(CHEMBL4576817)
Affinity DataIC50: 8.80nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531452BDBM50531452(CHEMBL4521489)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531434BDBM50531434(CHEMBL4458223)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50336977BDBM50336977(N-[5-(3-Fluoropyridin-4-yl)-6-pyridin-3-ylpyrazin-...)
Affinity DataKi:  24nMAssay Description:Inhibition of human A2B adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531477BDBM50531477(CHEMBL4448231)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531450BDBM50531450(CHEMBL4458042)
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531457BDBM50531457(CHEMBL4449139)
Affinity DataIC50: 42nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531451BDBM50531451(CHEMBL4462879)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531443BDBM50531443(CHEMBL4589448)
Affinity DataIC50: 55nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531437BDBM50531437(CHEMBL4474572)
Affinity DataIC50: 56nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 59nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at recombinant human A2B adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531444BDBM50531444(CHEMBL4564912)
Affinity DataIC50: 73nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531453BDBM50531453(CHEMBL4540250)
Affinity DataIC50: 97nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531463BDBM50531463(CHEMBL4516075)
Affinity DataIC50: 97nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531438BDBM50531438(CHEMBL4458469)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531464BDBM50531464(CHEMBL4540909)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531439BDBM50531439(CHEMBL4442438)
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531465BDBM50531465(CHEMBL4441343)
Affinity DataIC50: 145nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531456BDBM50531456(CHEMBL4457476)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531476BDBM50531476(CHEMBL4538262)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531416BDBM50531416(CHEMBL4451942)
Affinity DataIC50: 180nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531416BDBM50531416(CHEMBL4451942)
Affinity DataIC50: 180nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531420BDBM50531420(CHEMBL4553423)
Affinity DataIC50: 190nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531471BDBM50531471(CHEMBL4459477)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531449BDBM50531449(CHEMBL4522738)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531433BDBM50531433(CHEMBL4450633)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531448BDBM50531448(CHEMBL4452532)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531423BDBM50531423(CHEMBL4540558)
Affinity DataIC50: 210nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531454BDBM50531454(CHEMBL4440686)
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531430BDBM50531430(CHEMBL4452799)
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531460BDBM50531460(CHEMBL4560841)
Affinity DataIC50: 260nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531418BDBM50531418(CHEMBL4537687)
Affinity DataIC50: 280nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Rat)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at recombinant rat A2B adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531440BDBM50531440(CHEMBL4528081)
Affinity DataIC50: 300nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531470BDBM50531470(CHEMBL4453228)
Affinity DataIC50: 390nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531432BDBM50531432(CHEMBL4536104)
Affinity DataIC50: 390nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Mouse)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at recombinant mouse A2B adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531417BDBM50531417(CHEMBL4446433)
Affinity DataIC50: 430nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531467BDBM50531467(CHEMBL4569387)
Affinity DataIC50: 440nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531472BDBM50531472(CHEMBL4475483)
Affinity DataIC50: 440nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Mouse)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 470nMAssay Description:Antagonist activity at recombinant mouse A2A adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531441BDBM50531441(CHEMBL4543255)
Affinity DataIC50: 480nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531455BDBM50531455(CHEMBL4475461)
Affinity DataIC50: 490nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531436BDBM50531436(CHEMBL4541543)
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531424BDBM50531424(CHEMBL4585015)
Affinity DataIC50: 640nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at recombinant rat A2A adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531468BDBM50531468(CHEMBL4544040)
Affinity DataIC50: 760nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
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