Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50010259
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536919(CHEMBL4550236)
Affinity DataKi:  0.870nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataKi:  12nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as [35S]GTPgammaS binding after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536919(CHEMBL4550236)
Affinity DataKi:  12nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536913(CHEMBL4517991)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536904(CHEMBL4519981)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536903(CHEMBL4550003)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as [35S]GTPgammaS binding after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50380892(S-777469 | CHEMBL2019090)
Affinity DataKi:  36nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536903(CHEMBL4550003)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50006250(CHEMBL3139186)
Affinity DataKi:  40nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536913(CHEMBL4517991)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as [35S]GTPgammaS binding after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536906(CHEMBL4581598)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as [35S]GTPgammaS binding after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536906(CHEMBL4581598)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536921(CHEMBL4574224)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536904(CHEMBL4519981)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as [35S]GTPgammaS binding after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536914(CHEMBL4538593)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536911(CHEMBL4539849)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536910(CHEMBL4533329)
Affinity DataKi:  272nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536912(CHEMBL4518631)
Affinity DataKi:  281nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536901(CHEMBL4571345)
Affinity DataKi:  344nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536920(CHEMBL4516391)
Affinity DataKi:  438nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536915(CHEMBL4542489)
Affinity DataKi:  506nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536905(CHEMBL4548364)
Affinity DataKi:  526nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536921(CHEMBL4574224)
Affinity DataKi:  593nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536913(CHEMBL4517991)
Affinity DataKi:  627nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536904(CHEMBL4519981)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536903(CHEMBL4550003)
Affinity DataKi:  903nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataKi:  985nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536910(CHEMBL4533329)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536912(CHEMBL4518631)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536923(CHEMBL4565332)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536922(CHEMBL4585561)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536909(CHEMBL4562588)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536908(CHEMBL4586935)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536907(CHEMBL4514301)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536914(CHEMBL4538593)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50006250(CHEMBL3139186)
Affinity DataKi: >1.00E+3nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536918(CHEMBL4536203)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536902(CHEMBL4578601)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536901(CHEMBL4571345)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536917(CHEMBL4513395)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536911(CHEMBL4539849)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536906(CHEMBL4581598)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50536916(CHEMBL4575258)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50380892(S-777469 | CHEMBL2019090)
Affinity DataKi:  4.61E+3nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed