Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50009192
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009575BDBM50009575(CHEMBL3234446)
Affinity DataIC50: 0.0250nMAssay Description:Displacement of [125I]-(Glp1,Nle11,Try14)apelin-13 from recombinant rat EGFP-fused apelin receptor expressed in CHO cell membrane measured after 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009575BDBM50009575(CHEMBL3234446)
Affinity DataEC50:  1.90nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50525999BDBM50525999(CHEMBL4472749)
Affinity DataEC50:  2.5nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526001BDBM50526001(CHEMBL4550078)
Affinity DataEC50:  2.60nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257229BDBM50257229(CHEMBL4098390)
Affinity DataEC50:  4.10nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257231BDBM50257231(CHEMBL4065973)
Affinity DataEC50:  4.90nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526004BDBM50526004(CHEMBL4464954)
Affinity DataEC50:  6.30nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526000BDBM50526000(CHEMBL4440817)
Affinity DataEC50:  11nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526003BDBM50526003(CHEMBL4439951)
Affinity DataEC50:  176nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526002BDBM50526002(CHEMBL4559795)
Affinity DataEC50:  568nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed