Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50008945
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523811BDBM50523811(DNDI1416941 | CHEMBL2094331)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8296BDBM8296(CHEMBL102714 | cid_176158 | 3-(2,4-dichlorophenyl)...)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523808BDBM50523808(CHEMBL4474153)
Affinity DataIC50: 155nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523803BDBM50523803(CHEMBL4450851)
Affinity DataIC50: 233nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523807BDBM50523807(CHEMBL4514599)
Affinity DataIC50: 348nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523826BDBM50523826(CHEMBL4440139)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523805BDBM50523805(CHEMBL4529655)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523837BDBM50523837(CHEMBL4454916)
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50431816BDBM50431816(CHEMBL2347073)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523814BDBM50523814(CHEMBL4578156)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523812BDBM50523812(CHEMBL4448193)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523813BDBM50523813(CHEMBL3633203)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523810BDBM50523810(CHEMBL4580857)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523809BDBM50523809(CHEMBL4537467)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523806BDBM50523806(CHEMBL4101711)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523804BDBM50523804(CHEMBL4467292)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523829BDBM50523829(CHEMBL4438406)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523830BDBM50523830(CHEMBL4469665)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523827BDBM50523827(CHEMBL4516094)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523828BDBM50523828(CHEMBL4442846)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523825BDBM50523825(CHEMBL4545169)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523823BDBM50523823(CHEMBL4464997)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523824BDBM50523824(CHEMBL4085946)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523821BDBM50523821(CHEMBL4586793)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523822BDBM50523822(CHEMBL4449604)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523819BDBM50523819(CHEMBL4549051)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523820BDBM50523820(CHEMBL4577668)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523817BDBM50523817(CHEMBL4452454)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523815BDBM50523815(CHEMBL4517715)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523816BDBM50523816(CHEMBL4451858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523838BDBM50523838(CHEMBL4520227)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523836BDBM50523836(CHEMBL4525020)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523835BDBM50523835(CHEMBL4544396)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523833BDBM50523833(CHEMBL4585682)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523834BDBM50523834(CHEMBL3360387)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523831BDBM50523831(CHEMBL4476606)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523818BDBM50523818(CHEMBL4436958)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lomonosov Moscow State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523832BDBM50523832(CHEMBL4465183)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed