Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50007486 Sort by
LigandPNGBDBM252850(US9464076, 2 | US9464076, 6 | US9464076, 4 | US946...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509887(CHEMBL4529098)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509886(CHEMBL4439744)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509881(CHEMBL4589996)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM252856(US9464076, 8)
Affinity DataIC50: 13nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509893(CHEMBL4464258)
Affinity DataIC50: 23nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509882(CHEMBL4472246)
Affinity DataIC50: 23nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM14754(CHEMBL19224 | 1-[(3,4-dimethoxyphenyl)methyl]-6,7-...)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant rat PDE10A expressed in Sf9 cells using cGMP/cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509890(CHEMBL4449458)
Affinity DataIC50: 44nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509888(CHEMBL4448177)
Affinity DataIC50: 47nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509883(CHEMBL4587529)
Affinity DataIC50: 62nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM14754(CHEMBL19224 | 1-[(3,4-dimethoxyphenyl)methyl]-6,7-...)
Affinity DataIC50: 97nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50509885(CHEMBL4463792)
Affinity DataIC50: 110nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509880(CHEMBL4582678)
Affinity DataIC50: 120nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509891(CHEMBL4531756)
Affinity DataIC50: 200nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509884(CHEMBL4465465)
Affinity DataIC50: 320nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509892(CHEMBL4542313)
Affinity DataIC50: 440nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509889(CHEMBL4453464)
Affinity DataIC50: 510nMAssay Description:Inhibition of human MOLT4 cell-derived PDE10A using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50509881(CHEMBL4589996)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human MOLT4 cell-derived PDE7 using [3H]cAMP as substrate measured after 2 hrs in presence of rolipram/milrinone by topcount methodMore data for this Ligand-Target Pair
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PubMed