Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50009022
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50331094BDBM50331094(4-(3-chloro-4-(3-cyclopropylureido)phenoxy)-7-meth...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524583BDBM50524583(CHEMBL4455006 | US10980809, Example 70)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524587BDBM50524587(CHEMBL4466426 | US10980809, Example 20)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524586BDBM50524586(CHEMBL4449250 | US10980809, Example 65)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524588BDBM50524588(CHEMBL4528373 | US10980809, Example 47)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524589BDBM50524589(CHEMBL4581503 | US10980809, Example 71)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524578BDBM50524578(CHEMBL4514617 | US10980809, Example 18)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524584BDBM50524584(CHEMBL4516513 | US10980809, Example 67)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524579BDBM50524579(CHEMBL4531859 | US10980809, Example 23)
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524580BDBM50524580(CHEMBL4435366 | US10980809, Example 78)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524581BDBM50524581(CHEMBL4472616 | US10980809, Example 79)
Affinity DataIC50: 11nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524585BDBM50524585(CHEMBL4470543 | US10980809, Example 25)
Affinity DataIC50: 31nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Beijing University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524582BDBM50524582(CHEMBL4461971 | US10980809, Example 73)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human N-terminal GST-tagged VEGFR2 cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using Ulight-JA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed