Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50008742
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521804BDBM50521804(CHEMBL4581035)
Affinity DataIC50: 19nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521806BDBM50521806(CHEMBL4449908)
Affinity DataIC50: 37nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521803BDBM50521803(CHEMBL4568624)
Affinity DataIC50: 82nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521799BDBM50521799(CHEMBL4459270)
Affinity DataIC50: 86nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521800BDBM50521800(CHEMBL4470688)
Affinity DataIC50: 89nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521805BDBM50521805(CHEMBL4436644)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521801BDBM50521801(CHEMBL4521306)
Affinity DataIC50: 150nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521802BDBM50521802(CHEMBL4465300)
Affinity DataIC50: 200nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA gyrase subunit A(Escherichia coli)
University of Leeds

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521807BDBM50521807(CHEMBL4577939)
Affinity DataIC50: 410nMAssay Description:Inhibition of Escherichia coli DNA gyrase(A2B2 tetramer) preincubated for 5 mins followed by ATP addition and measured once per minute for 20 to 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed