Found 14 Enz. Inhib. hit(s) with all data for entry = 50007369 
Affinity DataIC50: 5.30nMAssay Description:Reversible inhibition of FAM-labeled peptide binding to full-length human N-terminal GST-tagged BTK (2 to 659 residues) expressed in baculovirus infe...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Reversible inhibition of FAM-labeled peptide binding to full-length human N-terminal GST-tagged BTK (2 to 659 residues) expressed in baculovirus infe...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 12nMAssay Description:Reversible inhibition of FAM-labeled peptide binding to full-length human N-terminal GST-tagged BTK (2 to 659 residues) expressed in baculovirus infe...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Reversible inhibition of FAM-labeled peptide binding to full-length human N-terminal GST-tagged BTK C481S mutant (2 to 659 residues) expressed in bac...More data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Reversible inhibition of FAM-labeled peptide binding to full-length human N-terminal GST-tagged BTK (2 to 659 residues) expressed in baculovirus infe...More data for this Ligand-Target Pair
Affinity DataIC50: 165nMAssay Description:Inhibition of human full-length recombinant FYN using KVEKIGEGTYGVVYK as substrate measured after 40 mins in presence of [gamma-33P]-ATP by scintilla...More data for this Ligand-Target Pair
Affinity DataIC50: 227nMAssay Description:Inhibition of recombinant human N-terminal GST-fused TEC catalytic domain (359 to 631 residues) expressed in baculovirus expression system using biot...More data for this Ligand-Target Pair
Affinity DataIC50: 307nMAssay Description:Inhibition of recombinant human ITK (352 to 617 residues) using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tsinghua University
Curated by ChEMBL
Tsinghua University
Curated by ChEMBL
Affinity DataIC50: 903nMAssay Description:Inhibition of recombinant full-length human SRC using KVEKIGEGTYGVVYK as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillati...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Z'-lyte-la...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Z'-lyte-la...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human full-length recombinant YES using poly(Glu, Tyr) 4:1 as substrate measured after 40 mins in presence of [gamma-33P]-ATP by scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Reversible inhibition of sodium orthovanadate-stimulated BTK autophosphorylation at Tyr223 residues in human Ramos cells preincubated for 2 hrs follo...More data for this Ligand-Target Pair
Affinity DataEC50: 101nMAssay Description:Reversible inhibition of sodium orthovanadate-stimulated BTK autophosphorylation at Tyr223 residues in human Ramos cells preincubated for 2 hrs follo...More data for this Ligand-Target Pair
