Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50007376
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Antagonist activity at human AChR alpha3beta4 transfected in human HEK293 cells assessed as decrease in epibatidine-induced calcium influx incubated ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Antagonist activity at human AChR alpha3beta4 transfected in human HEK293 cells assessed as decrease in epibatidine-induced calcium influx incubated ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Antagonist activity at human AChR alpha4beta2 transfected in human HEK293 cells assessed as decrease in epibatidine-induced calcium influx incubated ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at human AChR alpha4beta2 transfected in human HEK293 cells assessed as decrease in epibatidine-induced calcium influx incubated ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:Antagonist activity at human AChR alpha7 transfected in rat GH3 cells assessed as decrease in epibatidine-induced calcium influx incubated for 1 hr b...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4.53E+4nMAssay Description:Antagonist activity at human AChR alpha7 transfected in rat GH3 cells assessed as decrease in epibatidine-induced calcium influx incubated for 1 hr b...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.45E+5nMAssay Description:Antagonist activity at human AChR alpha4beta2 transfected in human HEK293 cells assessed as decrease in epibatidine-induced calcium influx incubated ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
American University of Health Sciences
Curated by ChEMBL
American University of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.67E+5nMAssay Description:Antagonist activity at human AChR alpha3beta4 transfected in human HEK293 cells assessed as decrease in epibatidine-induced calcium influx incubated ...More data for this Ligand-Target Pair


