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Found 25 Enz. Inhib. hit(s) with all data for entry = 50008869
TargetCytochrome P450 1A2(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523018(CHEMBL4577659)
Affinity DataEC50:  426nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523019(CHEMBL4440715)
Affinity DataEC50:  64nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523020(CHEMBL4466171)
Affinity DataEC50:  5nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523021(CHEMBL4441437)
Affinity DataEC50:  29nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523022(CHEMBL4549349)
Affinity DataEC50:  720nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523023(CHEMBL4454946)
Affinity DataEC50:  86nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523024(CHEMBL4515029)
Affinity DataEC50:  27nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523025(CHEMBL4525262)
Affinity DataEC50:  27nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523026(CHEMBL4442686)
Affinity DataEC50:  2.46E+3nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523027(CHEMBL4466588)
Affinity DataEC50:  301nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523028(CHEMBL4456673)
Affinity DataEC50:  31nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523029(CHEMBL4450117)
Affinity DataEC50:  7nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523017(CHEMBL4583270)
Affinity DataEC50:  430nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523016(CHEMBL4441091)
Affinity DataEC50:  44nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523015(CHEMBL4465577)
Affinity DataEC50:  261nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50508029(CHEMBL4467856)
Affinity DataEC50:  89nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523014(CHEMBL4548931)
Affinity DataEC50:  6nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523012(CHEMBL4476507)
Affinity DataEC50:  69nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50523013(CHEMBL4458134)
Affinity DataEC50:  25nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed