Found 9 Enz. Inhib. hit(s) with all data for entry = 50008230 TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Isf College Of Pharmacy
Curated by ChEMBL
Isf College Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Inhibition of 5HT transporter (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Isf College Of Pharmacy
Curated by ChEMBL
Isf College Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of 5HT transporter (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of HIV1 3B Y181C mutant infected in human MT2 cells assessed as reduction in virus-induced cytopathogenicity after 3 days by BrightGlo luc...More data for this Ligand-Target Pair
Affinity DataIC50: 6.22E+3nMAssay Description:Inhibition of recombinant human COX2 assessed as decrease in PGE2 release after 10 mins by EIAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C/K103N double mutant infected in human MT4 cells assessed as reduction in virus-induced cytopathogenici...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DHFRMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+5nMAssay Description:Inhibition of human DHFRMore data for this Ligand-Target Pair
