Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50007388
TargetSerine/threonine-protein kinase LATS2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild-type human partial length LATS2 (Q641 to V1088 residues) expressed in mammalian expression system assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MST2 (2 to end residues) assessed as residual activity using myelin basic protein as substrate measured after 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full-length human MST1 assessed as residual activity using KKSRGDYMTMQIG as substrate measured after 40 mins in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase LATS1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50508990(CHEMBL4472294)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant human LATS1 (Q678 to V1130 residues) expressed in bacterial expression system assessed as dissociation constant by Ki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed