Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50009120
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM33322(pyridazinone, 2-9)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525608(CHEMBL4590984)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525612(CHEMBL4524213)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525605(CHEMBL4520644)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM26658(2-(2,4-dihydroxyphenyl)-3,5,7-trihydroxychromen-4-...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525615(CHEMBL4435912)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525610(CHEMBL174487)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM26658(2-(2,4-dihydroxyphenyl)-3,5,7-trihydroxychromen-4-...)
Affinity DataIC50: 3.74E+4nMAssay Description:Inhibition of Staphylococcus aureus Newman recombinant SrtA expressed in Escherichia coli cells using Dabcyl-QALPETGEE-Edans as substrate by fluorime...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525613(CHEMBL4483668)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525607(CHEMBL4101630)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525609(CHEMBL4577169)
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525611(CHEMBL366787)
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525614(CHEMBL368170)
Affinity DataIC50: 5.21E+5nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSortase family protein(Staphylococcus aureus)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50525606(CHEMBL4470721)
Affinity DataIC50: 1.75E+6nMAssay Description:Inhibition of recombinant Staphylococcus aureus wild type truncated C-terminal His6 tagged Srt A using Abz-Leu-Pro-Glu-Thr-Gly-Lys(Dnp)-NH2 as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed