Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50008440
TargetGlucagon-like peptide 1 receptor(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50393572(CHEMBL2158488)
Affinity DataEC50:  203nMAssay Description:Agonist activity at human GLP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCathepsin L2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519377(CHEMBL4438688)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human cathepsin V using Z-Phe-Arg-7-amido-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetCathepsin L2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519381(CHEMBL4462944)
Affinity DataIC50: 700nMAssay Description:Inhibition of recombinant human cathepsin V using Z-Phe-Arg-7-amido-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519372(CHEMBL2158411)
Affinity DataEC50:  847nMAssay Description:Agonist activity at human GLP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCathepsin L2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519378(CHEMBL4576261)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human cathepsin V using Z-Phe-Arg-7-amido-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519376(CHEMBL4583627)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519373(CHEMBL3593481)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519384(CHEMBL4537425)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519382(CHEMBL4464398)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519379(CHEMBL4576254)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519375(CHEMBL4520281)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of human topoisomerase 2 by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519376(CHEMBL4583627)
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of human topoisomerase 2 by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519374(CHEMBL4462061)
Affinity DataIC50: 3.33E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using 4-nitrophenyl alpha-D-glucopyranoside as substarte preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519383(CHEMBL4543696)
Affinity DataIC50: 1.21E+6nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using 4-nitrophenyl alpha-D-glucopyranoside as substarte preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Nagasaki International University

Curated by ChEMBL
LigandPNGBDBM50519380(CHEMBL4555601)
Affinity DataIC50: 1.56E+6nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using 4-nitrophenyl alpha-D-glucopyranoside as substarte preincubated for 10 mins followed by substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed