Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50006723
LigandChemical structure of BindingDB Monomer ID 50502744BDBM50502744(CHEMBL4524153)
Affinity DataKi:  0.160nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 159183BDBM159183(US9034866, 660)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 158743BDBM158743(US9034866, 218)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502746BDBM50502746(CHEMBL3941082)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502741BDBM50502741(CHEMBL4517096)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502745BDBM50502745(CHEMBL4444206)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158675BDBM158675(US9034866, 150)
Affinity DataKi:  0.800nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 158675BDBM158675(US9034866, 150)
Affinity DataKi:  0.900nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 159183BDBM159183(US9034866, 660)
Affinity DataKi:  0.900nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158654BDBM158654(US9034866, 129)
Affinity DataKi:  1nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158743BDBM158743(US9034866, 218)
Affinity DataKi:  1.70nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158533BDBM158533(US9034866, 8)
Affinity DataKi:  3.10nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502744BDBM50502744(CHEMBL4524153)
Affinity DataKi:  3.60nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 159182BDBM159182(US9034866, 659)
Affinity DataKi:  4.20nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 158533BDBM158533(US9034866, 8)
Affinity DataKi:  4.90nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 158654BDBM158654(US9034866, 129)
Affinity DataKi:  5.90nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158562BDBM158562(US9034866, 37)
Affinity DataKi:  10nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 158645BDBM158645(US9034866, 120)
Affinity DataKi:  14nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158662BDBM158662(US9034866, 137)
Affinity DataKi:  14nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 158562BDBM158562(US9034866, 37)
Affinity DataKi:  25nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502743BDBM50502743(CHEMBL4461552)
Affinity DataKi:  44nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502747BDBM50502747(CHEMBL4546659)
Affinity DataKi:  62nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50502742BDBM50502742(CHEMBL3978002)
Affinity DataKi:  65nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 158645BDBM158645(US9034866, 120)
Affinity DataKi: >250nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50502742BDBM50502742(CHEMBL3978002)
Affinity DataKi:  582nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50502747BDBM50502747(CHEMBL4546659)
Affinity DataKi:  634nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50502745BDBM50502745(CHEMBL4444206)
Affinity DataKi: >1.25E+3nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50502741BDBM50502741(CHEMBL4517096)
Affinity DataKi: >1.25E+3nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50502743BDBM50502743(CHEMBL4461552)
Affinity DataKi: >1.25E+3nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 159182BDBM159182(US9034866, 659)
Affinity DataKi: >1.25E+3nMAssay Description:Inhibition of NIK (unknown origin) using ATP as substrate by transcreener ADP assay based fluorescence correlation spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed