Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50007923
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514023BDBM50514023(CHEMBL4447149)
Affinity DataIC50: 320nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514020BDBM50514020(CHEMBL4556236)
Affinity DataIC50: 930nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514028BDBM50514028(CHEMBL4474416)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514022BDBM50514022(CHEMBL4582907)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514016BDBM50514016(CHEMBL4524481)
Affinity DataIC50: 2.48E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514017BDBM50514017(CHEMBL4463336)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50400094BDBM50400094(CHEMBL427092)
Affinity DataIC50: 3.08E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514031BDBM50514031(CHEMBL4471787)
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514027BDBM50514027(CHEMBL4436783)
Affinity DataIC50: 4.56E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514026BDBM50514026(CHEMBL4585779)
Affinity DataIC50: 7.32E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514024BDBM50514024(CHEMBL4538482)
Affinity DataIC50: 8.53E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514029BDBM50514029(CHEMBL4532078)
Affinity DataIC50: 9.84E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514030BDBM50514030(CHEMBL4532373)
Affinity DataIC50: 9.84E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514019BDBM50514019(CHEMBL4514880)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514021BDBM50514021(CHEMBL4459452)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514018BDBM50514018(CHEMBL4517735)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514025BDBM50514025(CHEMBL4437373)
Affinity DataIC50: 5.57E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in hypoxia-induced human HCCLM3 cells co-transfected with luciferase reporter plasmid containing fiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed