Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50008265
TargetD(2) dopamine receptor(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517230(CHEMBL4467984)
Affinity DataKi:  0.840nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517232(CHEMBL4546839)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517229(CHEMBL4541515)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517236(CHEMBL4465127)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517222(CHEMBL4579585)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517233(CHEMBL4568756)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517221(CHEMBL4554135)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517223(CHEMBL4471116)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50010289((S)6-(Phenethyl-propyl-amino)-5,6,7,8-tetrahydro-n...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H] spiperone from human D2 dopamine receptor expressed in monkey caudate-putamen membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517226(CHEMBL4449666)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517227(CHEMBL4562705)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517225(CHEMBL4453578)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517224(CHEMBL4443273)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517234(CHEMBL4446228)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517235(CHEMBL4444520)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517231(CHEMBL4517197)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517228(CHEMBL4461338)
Affinity DataKi:  2.11E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed