Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with all data for entry = 50008527
TargetTubulin beta chain(Sus scrofa)
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50520178(CHEMBL4468642)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured at 30 secs interval for 65 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTubulin beta chain(Sus scrofa)
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKd:  1.13E+4nMAssay Description:Binding affinity to porcine brain tubulin polymerization by surface plasmon analysis analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50520178(CHEMBL4468642)
Affinity DataKd:  2.66E+3nMAssay Description:Binding affinity to porcine brain tubulin polymerization by surface plasmon analysis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB