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Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50018451
TargetAldehyde oxidase(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human liver AOX using phthalazine as substrate incubated for 2.5 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAldehyde oxidase(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50187243(17-ethinyl-3,17-estradiol | 17-ethinyl-3,17-oestra...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human liver AOX using phthalazine as substrate incubated for 2.5 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAldehyde oxidase(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human liver AOX using phthalazine as substrate incubated for 2.5 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAldehyde oxidase(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of human AOX using phthalazine as substrate preincubated for 30 mins followed by substrate addition by HPLC-MS analysisMore data for this Ligand-Target Pair
TargetAldehyde oxidase(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50130273(2-(4-[3-(2-chloro-10H-phenothiazin-10-yl)propyl]-1...)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of human liver AOX using phthalazine as substrate incubated for 2.5 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAldehyde oxidase(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of human liver AOX using phthalazine as substrate incubated for 2.5 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed