Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50011112
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544988(CHEMBL488823)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544983(CHEMBL4643934)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544984(CHEMBL4634233)
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544981(CHEMBL4649793)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544982(CHEMBL4636050)
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544986(CHEMBL4639190)
Affinity DataIC50: 2.98E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544985(CHEMBL4641564)
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544998(CHEMBL4639758)
Affinity DataIC50: 3.52E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544990(CHEMBL4649372)
Affinity DataIC50: 4.32E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544993(CHEMBL4641361)
Affinity DataIC50: 4.85E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544991(CHEMBL4643594)
Affinity DataIC50: 5.58E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544996(CHEMBL4632676)
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544989(CHEMBL4636870)
Affinity DataIC50: 5.91E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544995(CHEMBL4644329)
Affinity DataIC50: 5.96E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544999(CHEMBL4646705)
Affinity DataIC50: 6.27E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50244767(4-[[4-Oxo-2-thioxo-3-[3-(trifluoromethyl)phenyl]-5...)
Affinity DataIC50: 6.39E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544992(CHEMBL4647571)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50545000(CHEMBL4647496)
Affinity DataIC50: 7.63E+3nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544987(CHEMBL4642387)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544997(CHEMBL4641183)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50544994(CHEMBL4646548)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome (unknown origin) activation in LPS-primed bone marrow derived macrophage cells assessed as effect on IL-1beta produc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed