Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50010712
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541408(CHEMBL4643140)
Affinity DataKi:  0.00400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541406(CHEMBL4649325)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM362044(US10272077, Example 4 | US9833448, Example 4)
Affinity DataKi:  0.0150nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541407(CHEMBL4638635)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM391726(N-[(2R)-3-(7-methyl-1H- | US10300056, Example 11 |...)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM361594(US10272077, Example 1 | US9833448, Example 1)
Affinity DataKi:  0.0670nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541405(CHEMBL4633407)
Affinity DataKi:  0.110nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541410(CHEMBL4637301)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541413(CHEMBL4649671)
Affinity DataKi:  0.25nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50224431(CHEMBL236593 | MK-0974 | N-[(3R,6S)-6-(2,3-difluor...)
Affinity DataKi:  0.770nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541400(CHEMBL4634646)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541411(CHEMBL4643006)
Affinity DataIC50:  0.0100nMAssay Description:Inhibition of human CLR/RAMP1 by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50184069(CHEMBL207197 | N-((R)-1-((S)-6-amino-1-oxo-1-(4-(p...)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541409(CHEMBL4647045)
Affinity DataIC50:  0.0450nMAssay Description:Inhibition of human CLR/RAMP1 by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541412(CHEMBL4644508)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541404(CHEMBL4639133)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50047356(CHEMBL3334624)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541403(CHEMBL4641806)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50047357(CHEMBL3334623)
Affinity DataIC50:  44nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541402(CHEMBL4645875)
Affinity DataIC50:  250nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50541401(CHEMBL4634626)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 1(Homo sapiens (Human))
Biohaven Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173483((S)-6-Amino-2-[(R)-3-(3,5-dibromo-4-hydroxy-phenyl...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed