Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50007986
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246899BDBM50246899(N-{[(1S)-1-carboxy-5-{[(4-iodophenyl)carbonyl]amin...)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514660BDBM50514660(Dcfpyl | US10894807, ID P002)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514665BDBM50514665(CHEMBL4590944)
Affinity DataIC50: 4nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514657BDBM50514657(CHEMBL4461865)
Affinity DataIC50: 11nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514656BDBM50514656(CHEMBL4513630)
Affinity DataIC50: 12nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514650BDBM50514650(CHEMBL4445179)
Affinity DataIC50: 17nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514655BDBM50514655(CHEMBL4471968)
Affinity DataIC50: 107nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514658BDBM50514658(CHEMBL4466904)
Affinity DataIC50: 155nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514662BDBM50514662(CHEMBL4558538)
Affinity DataIC50: 195nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514654BDBM50514654(CHEMBL4586744)
Affinity DataIC50: 284nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514663BDBM50514663(CHEMBL4457563)
Affinity DataIC50: 399nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514661BDBM50514661(CHEMBL4453028)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514659BDBM50514659(CHEMBL4550529)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514653BDBM50514653(CHEMBL4514701)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514666BDBM50514666(CHEMBL4459899)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514651BDBM50514651(CHEMBL4439962)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514667BDBM50514667(CHEMBL4588782)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514652BDBM50514652(CHEMBL4524986)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514664BDBM50514664(CHEMBL4459755)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed