Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50007986
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50246899(N-{[(1S)-1-carboxy-5-{[(4-iodophenyl)carbonyl]amin...)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514660(Dcfpyl | US10894807, ID P002)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514665(CHEMBL4590944)
Affinity DataIC50: 4nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514657(CHEMBL4461865)
Affinity DataIC50: 11nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514656(CHEMBL4513630)
Affinity DataIC50: 12nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514650(CHEMBL4445179)
Affinity DataIC50: 17nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514655(CHEMBL4471968)
Affinity DataIC50: 107nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514658(CHEMBL4466904)
Affinity DataIC50: 155nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514662(CHEMBL4558538)
Affinity DataIC50: 195nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514654(CHEMBL4586744)
Affinity DataIC50: 284nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514663(CHEMBL4457563)
Affinity DataIC50: 399nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514661(CHEMBL4453028)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514659(CHEMBL4550529)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514653(CHEMBL4514701)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514666(CHEMBL4459899)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514651(CHEMBL4439962)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514667(CHEMBL4588782)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514652(CHEMBL4524986)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50514664(CHEMBL4459755)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PSMA in human LNCaP cell extracts in presence of N-acetylaspartylglutamate by Amplex red glutamic acid dependent fluorescence-based NAA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed