Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50009331
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)

Curated by ChEMBL
LigandPNGBDBM50527390(CHEMBL1232738)
Affinity DataKd:  320nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)

Curated by ChEMBL
LigandPNGBDBM50527390(CHEMBL1232738)
Affinity DataKd:  810nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)

Curated by ChEMBL
LigandPNGBDBM50240510(CHEMBL898 | DIFLUNISAL)
Affinity DataKd:  2.70E+3nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)

Curated by ChEMBL
LigandPNGBDBM50197883(CHEBI:78538 | FX-1006 | Tafamidis | US10377729, Co...)
Affinity DataKd:  1.05E+3nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)

Curated by ChEMBL
LigandPNGBDBM50197883(CHEBI:78538 | FX-1006 | Tafamidis | US10377729, Co...)
Affinity DataKd:  2.80E+3nMAssay Description:Stabilization of wild type human transthyretin expressed in Escherichia coli BL21(DE3) Star assessed as dissociation constant for TTR-amyloid beta (1...More data for this Ligand-Target Pair