Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50011173
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545428BDBM50545428(CHEMBL4648828)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545430BDBM50545430(CHEMBL4645823)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545429BDBM50545429(CHEMBL4641373)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545426BDBM50545426(CHEMBL4642262)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545427BDBM50545427(CHEMBL4637032)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545425BDBM50545425(CHEMBL4642172)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545420BDBM50545420(CHEMBL4640132)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545424BDBM50545424(CHEMBL4635366)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545434BDBM50545434(CHEMBL4648171)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545432BDBM50545432(CHEMBL4632739)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545423BDBM50545423(CHEMBL4637680)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545418BDBM50545418(CHEMBL4648880)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545425BDBM50545425(CHEMBL4642172)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545431BDBM50545431(CHEMBL4637897)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545419BDBM50545419(CHEMBL4641290)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545422BDBM50545422(CHEMBL4646402)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545430BDBM50545430(CHEMBL4645823)
Affinity DataKi:  296nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545432BDBM50545432(CHEMBL4632739)
Affinity DataKi:  336nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545433BDBM50545433(CHEMBL4642686)
Affinity DataKi:  355nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545418BDBM50545418(CHEMBL4648880)
Affinity DataKi:  363nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545433BDBM50545433(CHEMBL4642686)
Affinity DataKi:  364nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545420BDBM50545420(CHEMBL4640132)
Affinity DataKi:  365nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545424BDBM50545424(CHEMBL4635366)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545423BDBM50545423(CHEMBL4637680)
Affinity DataKi:  382nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545432BDBM50545432(CHEMBL4632739)
Affinity DataKi:  495nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545434BDBM50545434(CHEMBL4648171)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545422BDBM50545422(CHEMBL4646402)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545426BDBM50545426(CHEMBL4642262)
Affinity DataKi:  556nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545431BDBM50545431(CHEMBL4637897)
Affinity DataKi:  571nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545428BDBM50545428(CHEMBL4648828)
Affinity DataKi:  586nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545429BDBM50545429(CHEMBL4641373)
Affinity DataKi:  614nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545427BDBM50545427(CHEMBL4637032)
Affinity DataKi:  663nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545431BDBM50545431(CHEMBL4637897)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545419BDBM50545419(CHEMBL4641290)
Affinity DataKi:  874nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545430BDBM50545430(CHEMBL4645823)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545428BDBM50545428(CHEMBL4648828)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545429BDBM50545429(CHEMBL4641373)
Affinity DataKi:  1.17E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545423BDBM50545423(CHEMBL4637680)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545433BDBM50545433(CHEMBL4642686)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545426BDBM50545426(CHEMBL4642262)
Affinity DataKi:  2.45E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545427BDBM50545427(CHEMBL4637032)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545425BDBM50545425(CHEMBL4642172)
Affinity DataKi:  3.37E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545419BDBM50545419(CHEMBL4641290)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545422BDBM50545422(CHEMBL4646402)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545421BDBM50545421(CHEMBL4637391)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545424BDBM50545424(CHEMBL4635366)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545434BDBM50545434(CHEMBL4648171)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545418BDBM50545418(CHEMBL4648880)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545420BDBM50545420(CHEMBL4640132)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50545421BDBM50545421(CHEMBL4637391)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
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