TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Norman Drug Discovery Training And Consulting
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human BSEP expressed in HEK293 cell membrane vesicles assessed as reduction in 3H-TCA uptake incubated for 5 mins by radiodetection met...More data for this Ligand-Target Pair