Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50012815
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50428286(DABRAFENIB | GSK2118436A)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560548(CHEMBL4795335)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560555(CHEMBL4745503)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560559(CHEMBL4753878)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560547(CHEMBL4782235)
Affinity DataIC50:  11nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560557(CHEMBL4791677)
Affinity DataIC50:  13nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560546(CHEMBL4781905)
Affinity DataIC50:  14nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560554(CHEMBL4745087)
Affinity DataIC50:  17nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560549(CHEMBL4763209)
Affinity DataIC50:  20nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560553(CHEMBL4756122)
Affinity DataIC50:  23nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560560(CHEMBL4752201)
Affinity DataIC50:  25nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560550(CHEMBL4793770)
Affinity DataIC50:  28nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...)
Affinity DataIC50:  31nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560551(CHEMBL4762191)
Affinity DataIC50:  59nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560558(CHEMBL4755694)
Affinity DataIC50:  74nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560552(CHEMBL4746223)
Affinity DataIC50:  141nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50560556(CHEMBL4763983)
Affinity DataIC50:  152nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed