Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50012286
TargetHistamine H3 receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50247053(Tiprolisant | 1-(3-(3-(4-chlorophenyl)propoxy)prop...)
Affinity DataKi:  0.160nMAssay Description:Antagonist activity at recombinant human H3 receptor expressed in CHO-K1 cell membranes incubated for 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50556204(Lumateperone | ITI 007 | ITI-007 | ITI-722 | ITI00...)
Affinity DataIC50: 0.540nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50556204(Lumateperone | ITI 007 | ITI-007 | ITI-722 | ITI00...)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at postsynaptic D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50556204(Lumateperone | ITI 007 | ITI-007 | ITI-722 | ITI00...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of serotonin transporter (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50556204(Lumateperone | ITI 007 | ITI-007 | ITI-722 | ITI00...)
Affinity DataIC50: 4.10nMAssay Description:Partial agonist activity at presynaptic D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50556205(Darolutamide | Odm-201 | BAY 1841788 | BAY-1841788...)
Affinity DataKi:  11nMAssay Description:Inhibition of androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50177716(CHEMBL3813873 | US11679110, Compound Pexidartinib ...)
Affinity DataIC50: 20nMAssay Description:Inhibition of CSF1R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50556205(Darolutamide | Odm-201 | BAY 1841788 | BAY-1841788...)
Affinity DataIC50: 26nMAssay Description:Inhibition of androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataKi:  86nMAssay Description:Inhibition of androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50094975(US10053433, ARN-509 | ARN-509 | JNJ-56021927 | apa...)
Affinity DataKi:  93nMAssay Description:Inhibition of androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50094975(US10053433, ARN-509 | ARN-509 | JNJ-56021927 | apa...)
Affinity DataIC50: 200nMAssay Description:Inhibition of androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 219nMAssay Description:Inhibition of androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed