Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50013010
LigandChemical structure of BindingDB Monomer ID 14754BDBM14754(CHEMBL19224 | 1-[(3,4-dimethoxyphenyl)methyl]-6,7-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50058212BDBM50058212([9-(2-Fluoro-benzyl)-2-trifluoromethyl-9H-purin-6-...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 15296BDBM15296(Milrinone | CHEMBL189 | 6-methyl-2-oxo-5-pyridin-4...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant PDE3A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant PDE1B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50219334BDBM50219334(CHEMBL267102)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human recombinant PDE7A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human recombinant PDE1B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277784BDBM50277784(N,N,2-trimethyl-5-nitrobenzenesulfonamide | CHEMBL...)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of human recombinant PDE7A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562085BDBM50562085(CHEMBL4762789)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28393BDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of human recombinant PDE2A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562085BDBM50562085(CHEMBL4762789)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of human recombinant PDE5A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562105BDBM50562105(CHEMBL4755919)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 2.91E+3nMAssay Description:Inhibition of human recombinant PDE5A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562096BDBM50562096(CHEMBL4755193)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 3.53E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of human recombinant PDE4D using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50562098BDBM50562098(CHEMBL4781101)
Affinity DataIC50: 5.41E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562085BDBM50562085(CHEMBL4762789)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14363BDBM14363(5-(2-propoxyphenyl)-2H,3H,7H-[1,2,3]triazolo[4,5-d...)
Affinity DataIC50: 6.52E+3nMAssay Description:Inhibition of human recombinant PDE5A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 6.85E+3nMAssay Description:Inhibition of human recombinant PDE2A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562095BDBM50562095(CHEMBL4786151)
Affinity DataIC50: 7.09E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 7.24E+3nMAssay Description:Inhibition of human recombinant PDE7A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50059033BDBM50059033(CHEMBL71752 | cid_443955 | (11aS,11bS)-11a-Ethyl-2...)
Affinity DataIC50: 7.99E+3nMAssay Description:Inhibition of human recombinant PDE1B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562103BDBM50562103(CHEMBL4749066)
Affinity DataIC50: 8.34E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562085BDBM50562085(CHEMBL4762789)
Affinity DataIC50: 8.45E+3nMAssay Description:Inhibition of human recombinant PDE1B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562099BDBM50562099(CHEMBL4781432)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562087BDBM50562087(CHEMBL4789451)
Affinity DataIC50: 8.66E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562097BDBM50562097(CHEMBL4793395)
Affinity DataIC50: 9.77E+3nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 9.92E+3nMAssay Description:Inhibition of human recombinant PDE3A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 9.97E+3nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562107BDBM50562107(CHEMBL4778175)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562104BDBM50562104(CHEMBL4799953)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562088BDBM50562088(CHEMBL4752376)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562111BDBM50562111(CHEMBL4752998)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562106BDBM50562106(CHEMBL4764312)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562111BDBM50562111(CHEMBL4752998)
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of human recombinant PDE7A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562110BDBM50562110(CHEMBL4786766)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562108BDBM50562108(CHEMBL4798623)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of human recombinant PDE2A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562100BDBM50562100(CHEMBL4740026)
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562086BDBM50562086(CHEMBL4787162)
Affinity DataIC50: 2.58E+4nMAssay Description:Inhibition of human recombinant PDE4D using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 2.72E+4nMAssay Description:Inhibition of human recombinant PDE4D using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562092BDBM50562092(CHEMBL4758935)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 3.42E+4nMAssay Description:Inhibition of human recombinant PDE7A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562085BDBM50562085(CHEMBL4762789)
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of human recombinant PDE4D using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562089BDBM50562089(CHEMBL4798575)
Affinity DataIC50: 3.99E+4nMAssay Description:Inhibition of human recombinant PDE4B using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562084BDBM50562084(CHEMBL4784075)
Affinity DataIC50: 4.06E+4nMAssay Description:Inhibition of human recombinant PDE3A using cAMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50562085BDBM50562085(CHEMBL4762789)
Affinity DataIC50: 4.07E+4nMAssay Description:Inhibition of human recombinant PDE2A using cGMP as substrate incubated for 20 mins measured by Kinase Glo reagent based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
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