Affinity DataKi: 0.5nMAssay Description:Antagonist activity at human alphaVbeta3 Integrin assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human AchE by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human CXCR1More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human AchE by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human CXCR1More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human CXCR2-mediated chemotaxis expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of human BchE by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of Angiotensin 2 binding to Angiotensin 2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Angiotensin 2 binding to Angiotensin 2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Binding affinity to NMDA receptor (unknown origin)More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human CXCR1More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Binding affinity to NMDA receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human BchE by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Binding affinity to NMDA receptor (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Binding affinity to NMDA receptor (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity to TCP-stimulated NMDA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of MMP-1 (unknown origin) using DnpPro-Cha-Gly-Cys(Me)-His-Ala-Lys(Nma)-NH2 as substrate by fluorescence spectroscopyMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataKd: 0.0490nMAssay Description:Binding affinity to human CXCR2 assessed as dissociation constant incubated for 6 to 24 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Palacky University Olomouc
Curated by ChEMBL
Palacky University Olomouc
Curated by ChEMBL
Affinity DataKd: 3.90nMAssay Description:Binding affinity to human CXCR1 assessed as dissociation constant incubated for 6 to 24 hrs by radioligand binding assayMore data for this Ligand-Target Pair