Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50012333
TargetProteasome subunit beta type-5(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556643(CHEMBL4786009)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of chymotrypsin-like activity 20S proteasome beta subunit 5 of human MCF7 cells using fluorogenic substrate Suc-LLVY-AMC after 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556644(NSC-45382 | CHEMBL1214274)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of chymotrypsin-like activity 20S proteasome beta subunit 5 of human MCF7 cells using fluorogenic substrate Suc-LLVY-AMC after 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556643(CHEMBL4786009)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of trypsin-like activity 20S proteasome beta subunit 2 of human MCF7 cells using fluorogenic substrate Boc-LRR-AMC after 1 hr by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556644(NSC-45382 | CHEMBL1214274)
Affinity DataIC50: 2.64E+4nMAssay Description:Inhibition of trypsin-like activity 20S proteasome beta subunit 2 of human MCF7 cells using fluorogenic substrate Boc-LRR-AMC after 1 hr by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556645(CHEMBL4796470)
Affinity DataIC50: 3.31E+4nMAssay Description:Inhibition of chymotrypsin-like activity 20S proteasome beta subunit 5 of human MCF7 cells using fluorogenic substrate Suc-LLVY-AMC after 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556643(CHEMBL4786009)
Affinity DataIC50: 4.48E+4nMAssay Description:Inhibition of caspase-like activity 20S proteasome beta subunit 1 of human MCF7 cells using fluorogenic substrate Z-LLE-AMC after 1 hr by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556645(CHEMBL4796470)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of trypsin-like activity 20S proteasome beta subunit 2 of human MCF7 cells using fluorogenic substrate Boc-LRR-AMC after 1 hr by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556645(CHEMBL4796470)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of caspase-like activity 20S proteasome beta subunit 1 of human MCF7 cells using fluorogenic substrate Z-LLE-AMC after 1 hr by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Ege University

Curated by ChEMBL
LigandPNGBDBM50556644(NSC-45382 | CHEMBL1214274)
Affinity DataIC50: 5.31E+4nMAssay Description:Inhibition of caspase-like activity 20S proteasome beta subunit 1 of human MCF7 cells using fluorogenic substrate Z-LLE-AMC after 1 hr by fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed