Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50013809
TargetAndrogen receptor(Homo sapiens (Human))
Bc Cancer

Curated by ChEMBL
LigandPNGBDBM50569842(CHEMBL4871230)
Affinity DataIC50:  3.50E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells transfected with PSA assessed as inhibition of R1881-induced PSA luciferase activity pretreated with c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bc Cancer

Curated by ChEMBL
LigandPNGBDBM50569840(CHEMBL4852950)
Affinity DataIC50:  6.50E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells transfected with PSA assessed as inhibition of R1881-induced PSA luciferase activity pretreated with c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bc Cancer

Curated by ChEMBL
LigandPNGBDBM50569842(CHEMBL4871230)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of R1881-stimulated AR transcription driven human LNCaP cells proliferation preincubated for 1 hr followed by R1881 addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bc Cancer

Curated by ChEMBL
LigandPNGBDBM50569841(CHEMBL4861372)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at AR in human LNCaP cells transfected with PSA assessed as inhibition of R1881-induced PSA luciferase activity pretreated with c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bc Cancer

Curated by ChEMBL
LigandPNGBDBM50569841(CHEMBL4861372)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of R1881-stimulated AR transcription driven human LNCaP cells proliferation preincubated for 1 hr followed by R1881 addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bc Cancer

Curated by ChEMBL
LigandPNGBDBM50569840(CHEMBL4852950)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of R1881-stimulated AR transcription driven human LNCaP cells proliferation preincubated for 1 hr followed by R1881 addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed