Found 5 Enz. Inhib. hit(s) with all data for entry = 50016393 
Affinity DataKi: 400nMAssay Description:Competitive inhibition of p300 HAT domain (unknown origin) using varying concentrations of acetyl-CoA and constant concentration of H4-15 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of heat inactivated recombinant human HDAC6 expressed in HEK293T cells assessed as inhibition of tau protein deacetylation incubated for 1...More data for this Ligand-Target Pair
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Karolinska Institutet
Curated by ChEMBL
Karolinska Institutet
Curated by ChEMBL
Affinity DataIC50: 294nMAssay Description:Inhibition of recombinant polyhistidine-tagged human tau40 aggregation assessed as reduction in filament formation by measuring total filament length...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide GSM as substrate incubated for 30 mins in presence of ATP by Kinase-Glo ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of C-terminal His-tagged recombinant human BACE-1 expressed in mouse NSO cells using methoxy coumarin Ser-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-...More data for this Ligand-Target Pair
