Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50012342
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556717(CHEMBL4780703)
Affinity DataIC50: 630nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556698(CHEMBL2375494)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556715(CHEMBL4782344)
Affinity DataIC50: 880nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556716(CHEMBL4796964)
Affinity DataIC50: 910nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556721(CHEMBL4790746)
Affinity DataIC50: 1.01E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556719(CHEMBL4782590)
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556710(CHEMBL4741257)
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556706(CHEMBL4797370)
Affinity DataIC50: 1.49E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556718(CHEMBL4787771)
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556699(CHEMBL4746541)
Affinity DataIC50: 1.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556705(CHEMBL4793323)
Affinity DataIC50: 1.72E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556708(CHEMBL4795327)
Affinity DataIC50: 1.76E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556700(CHEMBL4761208)
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556722(CHEMBL4791780)
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556720(CHEMBL4745132)
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556709(CHEMBL4783011)
Affinity DataIC50: 2.37E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556703(CHEMBL4761078)
Affinity DataIC50: 2.57E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556701(CHEMBL4746014)
Affinity DataIC50: 2.63E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556702(CHEMBL4763588)
Affinity DataIC50: 2.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556704(CHEMBL4740701)
Affinity DataIC50: 3.02E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556713(CHEMBL4748854)
Affinity DataIC50: 3.29E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556714(CHEMBL4777734)
Affinity DataIC50: 3.54E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556707(CHEMBL4762863)
Affinity DataIC50: 3.87E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556723(CHEMBL240484)
Affinity DataIC50: 5.45E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556712(CHEMBL4798117)
Affinity DataIC50: 7.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetG-protein coupled receptor 52(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556711(CHEMBL4755423)
Affinity DataIC50: 8.13E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed