Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50012945
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516881(US11104665, Example 1.2)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516886(US11104665, Example 2.1)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516883(US11104665, Example 1.4)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516884(US11104665, Example 1.5)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516890(US11104665, Example 2.5)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516880(US11104665, Example 1.1)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516888(US11104665, Example 2.3)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human autotaxin assessed as reduction in LPA production using LPC as substrate after 2 hrs by Rapidfire-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516884(US11104665, Example 1.5)
Affinity DataIC50: 9nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516886(US11104665, Example 2.1)
Affinity DataIC50: 33nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516880(US11104665, Example 1.1)
Affinity DataIC50: 46nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516881(US11104665, Example 1.2)
Affinity DataIC50: 55nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516888(US11104665, Example 2.3)
Affinity DataIC50: 186nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516883(US11104665, Example 1.4)
Affinity DataIC50: 201nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAutotaxin(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM516890(US11104665, Example 2.5)
Affinity DataIC50: 264nMAssay Description:Inhibition of ATX in human whole blood assessed as reduction in LPA level after 1 hr by rapidFire based MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed